5A3T: Crystal structure of human PLU-1 (JARID1B) in complex with KDM5-C49 (2-(((2-((2-(dimethylamino)ethyl)(ethyl)amino)-2-oxo
Crystal structure of human PLU-1 (JARID1B) in complex with KDM5-C49 (2-(((2-((2-(dimethylamino)ethyl)(ethyl)amino)-2-oxoethyl)amino)methyl) isonicotinic acid).. Determined by x-ray diffraction at 1.9 Å resolution. Released 2015.
Composition
This structure contains 4,008 atoms across 1 protein chain. Molecular weight: 56.62 kDa.
Primary citation
Structural Analysis of Human Kdm5B Guides Histone Demethylase Inhibitor Development.. Johansson, C., Velupillai, S., Tumber, A. et al., Nat.Chem.Biol. (2016).
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