6U7C: Human GRK2 in complex with Gbetagamma subunits and CCG258747

Human GRK2 in complex with Gbetagamma subunits and CCG258747. Determined by x-ray diffraction at 2.44 Å resolution. Released 2020.

Composition

This structure contains 8,327 atoms across 3 protein chains. Molecular weight: 125.48 kDa.

Primary citation

A New Paroxetine-Based GRK2 Inhibitor Reduces Internalization of themu-Opioid Receptor.. Bouley, R.A., Weinberg, Z.Y., Waldschmidt, H.V. et al., Mol.Pharmacol. (2020).

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Source: RCSB Protein Data Bank